Anti-Aging & Longevity

Rapamycin

Also known as: Sirolimus · mTOR inhibitor

The only drug proven to extend lifespan in mammals — the gold standard longevity compound.

Half-Life
~62 hours
Administration
Oral
Category
Anti-Aging & Longevity
Citations
2 studies

What is Rapamycin?

Rapamycin (Sirolimus) is an mTOR (mechanistic target of rapamycin) inhibitor originally developed as an immunosuppressant for organ transplants. It is the only drug that has consistently extended lifespan in multiple mammalian species, including mice (up to 25% lifespan extension even when started in old age). It is used off-label by longevity researchers and physicians.

Mechanism of Action

Rapamycin inhibits mTORC1, the master regulator of cellular growth and metabolism. mTORC1 inhibition activates autophagy, reduces protein synthesis (reducing cellular 'noise'), improves mitochondrial function, reduces senescent cell accumulation, and mimics the effects of caloric restriction at the cellular level.

Rapamycin Dosing Protocol

Longevity protocol: 1–6 mg/week oral (intermittent dosing). Most longevity physicians use 2–5 mg/week or 1–2 mg/day for 2 days/week. Immunosuppressive doses (organ transplant): 2–5 mg/day — much higher than longevity doses. Blood level monitoring recommended.

Administration Routes
Oral
Half-Life
~62 hours

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Rapamycin Benefits

Proven lifespan extension in mammals (up to 25%)
Autophagy activation
Reduced cancer risk
Improved immune function (at low doses)
Reduced senescent cell accumulation
Cardiovascular protection
Neuroprotection

Side Effect Profile

At immunosuppressive doses: significant immune suppression, infection risk, metabolic effects. At longevity doses (1–6 mg/week): generally well-tolerated, but potential for mouth sores, mild immune effects, metabolic changes. Requires physician oversight and monitoring.

Rapamycin Stacking Guide

Rapamycin works synergistically with these compounds. Click any to learn more, or ask PepBot to build you a complete stack.

Research & Citations

Frequently Asked Questions about Rapamycin

Is Rapamycin safe for longevity use?
At low intermittent doses (1–6 mg/week), Rapamycin appears to be well-tolerated based on clinical experience from longevity physicians like Dr. Peter Attia and Dr. Matt Kaeberlein. The key is using longevity doses (not immunosuppressive doses) and monitoring with bloodwork. It requires a physician prescription and oversight — this is not a self-experiment compound.

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